Poster Session 2 and Drinks — ASN Events

Poster Session 2 and Drinks — ASN Events

Poster Session 2 and Drinks

Synthesis and application of advanced fluorescent probes (#165)

Alejandra Gallardo-Godoy

Detection of bioactive peptides including gonadotrophin-releasing factors (GnRHs) in horse urine using ultra-high performance liquid chromatography-high resolution mass spectrometry (UHPLC-HRMS) (#166)

Photooxidation of oxazoles – a new approach to solid-phase peptide synthesis (#167)

Chloe N. Larcombe

Development of novel relaxin-3 analogues for blood-brain barrier penetration (#168)

Phosphorylation of α-synuclein induces distinct strains and propagation properties (#169)

Dichloroacetone – A robust approach to acetone-linked bicyclic dimer peptides (#170)

Qingqing (Irene) Lin

Synthesis of Peptide Natural Products Enabled by New Strategies for Late-Stage Modification (#171)

The role of charge regulation in the interaction between oligo-peptides and polyelectrolytes (#172)

Insulin fatty acid acylation scan: Discovery of Insulin 327, an acylated hepato-preferential insulin analogue with high insulin receptor affinity (#173)

Robust methodology for assembling peptides with tryptophan C-mannosylation (#174)

Peptide modulating tension in cell membranes: the regulation of cell movement and morphology via actin remodeling (#175)

Toshihiro Masuda

Tyrosine sulfation is an important post-translational modification in anti-inflammatory peptides from blood-feeding organisms. (#177)

Joshua W Maxwell

The New Kid On The Block: Discovery and development of Na_V channel inhibitor and µ-conotoxin NgIIIA (#178)

Kirsten L McMahon

Peptide cyclisation using a pyridine-2,6-dicarbonitrile linker (#179)

Richard Morewood

Structure-activity study of the analgesic NaV1.7 inhibiting venom peptide Pn3a (#180)

Alexander Mueller

Chemical strategies to tune potency, selectivity and stability of neuropeptides (#181)

Markus Muttenthaler

Design and synthesis of a PD-1 binding peptide and evaluation of its anti-tumor activity (#182)

A Zn(II)-catalyst permits bis-thioether peptide stapling under non-basic conditions (#183)

Noncanonical peptides as probes and inhibitors for flavivirus proteases (#184)

Christoph Nitsche

Identification and Optimisation of a Lead Bromodomain Inhibitor (#185)

Alexander R Norman

Membrane-bound structure and membrane selectivity of cationic antimicrobial peptide Hymenochirin-1Pa and its D9K analog (#186)

Evaluation of biological activity of frog skin-derived peptide, ranatensin (#187)

Liliana Mrs. Palczynska

Thiol-cyanobenzothiazole ligation: an efficient preparation of peptide-oligonucleotide conjugates (#188)

The Structural Features of an Ancient Peptide Family Buried within Vicilin Precursors. (#189)

Colton D. Payne

Cyclic peptide conjugates: their mode-of action and interaction with cell membranes (#190)

Gregoire Philippe

Cyclic peptides to probe the internal interactome of PDZ domains (#192)

Javier Rodriguez Balboa

Decoding the complex regulation of cone snail venoms: connecting evolution and drug discovery (#193)

Novel methods for inhibiting amyloidogenesis in the presence of peptides in order to block hydrophobic interaction (#194)

Masatoshi Saiki

Cytosolic Delivery of Macromolecules by Endosomolytic Cationic Helical Peptide (#195)

Kentarou Sakamoto

Exploring the oxytocin receptor as a novel target for breast cancer (#196)

Cristina Sanchez de la Rosa

Affinity-based functionalization of biomedical polymeric micelles through polymer-binding peptides (#197)

Backbone cyclization of native α-conotoxin CIA: Influences on structure and bioactivity (#198)

The use of peptide-membrane interactions in the design of selective and potent sodium channel inhibitors (#199)

Christina Schroeder

Discovery of tight binding inhibitors of hip1 a mycobacterium tuberculosis drug target (#200)

Nicholas C Schuman

Conformational diversity in the neurotensin peptide upon binding neurotensin receptor 1 may drive receptor activation (#201)

Discovery and mechanistic investigations of ultrashort amphiphilic peptides that exhibit potent inhibition of Cryptococcus neoformans (#202)

Tripeptide-induced mechanical property modulation of mesenchymal stem cells stimulates proliferation and wound healing (#203)

Enhancing activity by combining antimicrobial peptides and antibiotics (#204)

Evolving Peptide G Protein-Coupled Receptors (GPCRs) to Facilitate Structural Studies Using a Novel Lentiviral Based Method of Directed Evolution (#205)

Peptide based hydrogen sulfide responsive nanostructures for biomedical applications (#206)

Analysis of granulin peptide folding (#207)

Synthesis and biological activity of celogentin analogues (#208)

Varsha Thombare

Iterative optimization of the cyclic peptide SFTI-1 yields potent inhibitors of neutrophil proteinase 3 (#209)

Taking active steps to improving the pharmacokinetics of disulfide-rich peptides (#210)

Benjamin J Tombling

μ‐Conotoxin KIIIA isomer selectivity on human voltage gated sodium channels (#211)

Enzymatic ligation of Na_v1.7-inhibiting gating modifier and pore blocker toxins (#212)

Exploration of amyloidogenic core β-sheet and the FEL-mediated dissociation of amyloid fibrils in SAA (#213)

The characterization of triglyceride-based nanodroplets and their interaction with lipid specific peptides and proteins (#214)

Valerija Vezočnik

A fluorescent protein-tagged peptide toxin as a tool for K_V1.3 visualisation (#215)

Combinatorial peptide libraries in venoms of Australian nettle caterpillars (#216)

Andrew A Walker

From sunflower to skin cancer: Development of melanocortin receptor-1 agonists based on the cyclic peptide framework of sunflower trypsin inhibitor-1 (#217)

Development of a lentiviral nanobody screening platform against peptide GPCRs (#218)

Lisa M Williams

Delivery of a peptide-based vaccine against Group A Streptococcus with the help of cell penetrating peptides (#219)

Anchoring epitopes to improve grafted peptide structure and activity (#220)

A*STAR Peptide Engineering Platform (PEP): Targeting Macrocyclic Modalities for Protein-Protein Interactions (#221)

In-cell structure determination of an antimicrobial peptide by DNP solid-state NMR (#222)

Peptidomimetics targeting the SOCS-SH2 domain (#223)

Receptor-Mediated MAPK and Akt Signaling are Maintained in Gamma-Irradiated FroZen Cells (#224)

Synthesis and Evaluation of a Library of Self-Adjuvanting Peptide and Protein Vaccines against Mycobacterium tuberculosis (#225)

Development of a single-chain peptide agonist for the G-protein-coupled receptor, RXFP1 (#226)

Praveen Praveen

Improving in vivo analgesia through glycosylation of bilorphin, a biased μ-opioid derived from a novel tetrapeptide class found in an Australian fungus (#227)